General
Preferred name
C-82
Synonyms
P&D ID
PD162521
CAS
1422253-37-9
Tags
available
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
PRICE
1399
DESCRIPTION
C-82 is a specific CBP/??-catenin antagonist. It inhibits the binding between ??-catenin and CBP and increases the binding between ??-catenin and p300.
DESCRIPTION
C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and increases the binding between β-catenin and p300.
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
4
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
7
Molecular Weight
578.26
Hydrogen Bond Acceptors
6
Hydrogen Bond Donors
2
Rotatable Bonds
6
Ring Count
6
Aromatic Ring Count
4
cLogP
3.51
TPSA
109.32
Fraction CSP3
0.27
Chiral centers
3.0
Largest ring
6.0
QED
0.36
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Target
CBP
β-catenin
Wnt
Pathway
Chromatin/Epigenetic
Cytoskeletal Signaling
Stem Cells
Stem Cell/Wnt
Source data
