General
Preferred name
SULTAMICILLIN
Synonyms
Bacimex ()
Unacim orale ()
Unasyn ()
sultamycillin tosylate ()
Sultamicillin (tosylate) ()
Sultamicillin (tosilate) ()
Sultamicillin Tosylate ()
Sultamicillin Tosilate ()
Unacid ()
CP-49952 ()
CP-49,952 ()
VD-1827 ()
Sultamicilina ()
Sultamicilline ()
Sultamycillin ()
P&D ID
PD072126
CAS
76497-13-7
83105-70-8
Tags
available
prodrug
drug
Drug Status
approved
investigational
Max Phase
2.0
Drug indication
bacterial disease
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
DESCRIPTION
Sultamicillin is a prodrug of and linked as a double ester. This orally bioavailable molecule has similar antibacterial activity and clinical efficacy to that of the parenteral formulation of ampicillin and sulbactam .
(GtoPdb)
PRICE
29
DESCRIPTION
Sultamicillin is a broad-spectrum and orally active beta-lactamase inhibitor, an antibiotic with antibacterial activity[1].
DESCRIPTION
Sultamicillin is an orally active double prodrug of Ampicillin/Sulbactan. Sulbactam is a semisynthetic ??-Lactamase inhibitor.
PRICE
29
DESCRIPTION
Sultamicillin tosylate is a broad-spectrum and orally active beta-lactamase inhibitor, an antibiotic with antibacterial activity[1].
DESCRIPTION
Sultamicillin is an orally active double prodrug of Ampicillin/Sulbactan. Sulbactam is a semisynthetic β-Lactamase inhibitor.
(TargetMol Bioactive Compound Library)
DESCRIPTION
Sultamicillin Tosylate (Unacim orale) is an oral form of the antibiotic combination (codrug or mutual prodrug) ampicillin/sulbactam.
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
13
ChEMBL Drugs
CZ-OPENSCREEN Bioactive Library
Drug Repurposing Hub
DrugBank
DrugBank Approved Drugs
DrugCentral
DrugCentral Approved Drugs
Guide to Pharmacology
Natural product-based probes and drugs
ReFrame library
Selleckchem Bioactive Compound Library
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
42
Molecular Weight
594.15
Hydrogen Bond Acceptors
11
Hydrogen Bond Donors
2
Rotatable Bonds
7
Ring Count
5
Aromatic Ring Count
1
cLogP
-0.59
TPSA
182.48
Fraction CSP3
0.56
Chiral centers
6.0
Largest ring
6.0
QED
0.23
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Target
antibiotic
Bacterial
β-Lactamase
¦Â-Lactamase
MOA
Antibiotic inhibitor
antibacterial
Indication
gram-negative bacterial infections, gram-positive bacterial infections
Biosynthetic Origin
Peptide (beta-Lactam)
Therapeutic Indication
Antibacterial
Therapeutic Class
Antimicrobial
Pathway
Microbiology/virology
Anti-infection
Source data
