General
Preferred name
TABIMORELIN
Synonyms
Tabimorelin hemifumarate ()
NN-703 ()
Nn703 ()
NNC-26-0703 ()
Tabimoreline ()
Tabimorelina ()
P&D ID
PD070598
CAS
242143-80-2
193079-69-5
Tags
available
drug candidate
Drug indication
Growth hormone deficiency
Drug Status
investigational
Max Phase
2.0
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
DESCRIPTION
Highly potent NTS receptor antagonist
(Tocris Bioactive Compound Library)
DESCRIPTION
Potent, orally active ghrelin receptor agonist
(Tocriscreen Total)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Cell lines
0
Organisms
1
Compound Sets
8
ChEMBL Drugs
CZ-OPENSCREEN Bioactive Library
Drug Repurposing Hub
DrugMAP
LSP-MoA library (Laboratory of Systems Pharmacology)
ReFrame library
Tocris Bioactive Compound Library
Tocriscreen Total
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
25
Molecular Weight
528.31
Hydrogen Bond Acceptors
4
Hydrogen Bond Donors
2
Rotatable Bonds
11
Ring Count
3
Aromatic Ring Count
3
cLogP
3.71
TPSA
95.74
Fraction CSP3
0.34
Chiral centers
2.0
Largest ring
6.0
QED
0.37
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Primary Target
Ghrelin Receptors
MOA
Agonist
growth hormone secretagogue receptor agonist
Target
GHSR
Source data
