General
Preferred name
PILSICAINIDE
Synonyms
SUN 1165 ()
Pilsicainide hydrochloride ()
Pilsicainide (hydrochloride) ()
SUN-1165 ()
Pilzicainide(hydrochloride) ()
Pilsicainide HCl ()
Pilsicainida ()
P&D ID
PD013798
CAS
88069-67-4
88069-49-2
Tags
available
drug
Drug indication
Heart arrhythmia
Drug Status
approved
investigational
Max Phase
2.0
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
DESCRIPTION
Pilsicainide hydrochloride (SUN-1165) is an orally active sodium channel blocker and potent class Ic antiarrhythmic agent[1][2].
PRICE
29
DESCRIPTION
Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
13
Cayman Chemical Bioactives
ChEMBL Drugs
Drug Repurposing Hub
DrugBank
DrugCentral
DrugCentral Approved Drugs
DrugMAP
DrugMAP Approved Drugs
DrugMatrix
MedChem Express Bioactive Compound Library
NPC Screening Collection
ReFrame library
TargetMol Bioactive Compound Library
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
38
Molecular Weight
272.19
Hydrogen Bond Acceptors
2
Hydrogen Bond Donors
1
Rotatable Bonds
3
Ring Count
3
Aromatic Ring Count
1
cLogP
3.26
TPSA
32.34
Fraction CSP3
0.59
Chiral centers
0.0
Largest ring
6.0
QED
0.92
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Target
Sodium Channel
SCN5A
Indication
cardiac arrythmia
MOA
Sodium Channel blocker
Pathway
Membrane Transporter/Ion Channel
Source data
