General
Preferred name
MEPTAZINOL
Synonyms
MEPTAZINOL HYDROCHLORIDE ()
Riemser brand of meptazinol hydrochloride ()
Meptazinol HCl ()
WY-22811 HYDROCHLORIDE ()
Meptid ()
IL-22811 HCL ()
WY-22811 HCL ()
IL 22811 HCL ()
IL-22811 HYDROCHLORIDE ()
WY 22811 HCL ()
WY-22811 ()
IL-22811 ()
Meptazinol (hydrochloride) ()
P&D ID
PD013172
CAS
59263-76-2
54340-58-8
Tags
available
drug candidate
drug
First approval
1983
Drug indication
Pain
Drug Status
approved
experimental
investigational
Max Phase
2.0
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
PRICE
41
DESCRIPTION
Meptazinol is an opioid receptor agonist, with analgesic action. The INN recprod for this drug shows that it is a mixture of enantiomers. We show the molecule without specified stereochemistry to represent the mixture.
(GtoPdb)
DESCRIPTION
mu1 partial agonist
(Tocriscreen Plus)
DESCRIPTION
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
14
Cayman Chemical Bioactives
ChEMBL Drugs
DrugBank
DrugCentral
DrugCentral Approved Drugs
DrugMAP
DrugMAP Approved Drugs
DrugMatrix
Guide to Pharmacology
NPC Screening Collection
Prestwick Chemical Library
ReFrame library
TargetMol Bioactive Compound Library
Tocriscreen Plus
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
44
Molecular Weight
233.18
Hydrogen Bond Acceptors
2
Hydrogen Bond Donors
1
Rotatable Bonds
2
Ring Count
2
Aromatic Ring Count
1
cLogP
3.16
TPSA
23.47
Fraction CSP3
0.6
Chiral centers
1.0
Largest ring
7.0
QED
0.85
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Target Type
7-TM Receptors
Target
Opioid Receptor
Pathway
Endocrinology/Hormones
GPCR/G protein
Neuroscience
Source data
