General
Preferred name
AZACYCLONOL
Synonyms
¦Ã-pipradol ()
Diphenyl-piperidin-4-yl-methanol ()
Ataractan ()
γ-pipradol ()
MDL 4829 ()
MER 17 ()
??pipradol ()
Diphenyl(piperidin-4-yl)methanol ()
MER 17, MDL 4829 ()
AZACYCLONOL HYDROCHLORIDE ()
Calmeran ()
Psychosan ()
gamma-Pipradol ()
Frenoton ()
Azaciclonol ()
Azacyclonol hcl ()
Frenquel ()
P&D ID
PD010763
CAS
115-46-8
1798-50-1
Tags
available
drug
drug candidate
Drug indication
Discovery agent
Drug Status
approved
investigational
Max Phase
2.0
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
DESCRIPTION
Azacyclonol (¦Ã-pipradol), a metabolite of Terfenadine, is a central depressant agent. Azacyclonol is a ganglion-blocking agent. Azacyclonol can be used to diminish psychoses-induced hallucinations[1][2][3].
PRICE
29
DESCRIPTION
Azacyclonol, also known as γ-pipradol, is a drug used to diminish hallucinations in psychotic individuals.
(BOC Sciences Bioactive Compounds)
DESCRIPTION
Azacyclonol is a CNS depressant, used to diminish hallucinations in psychotic individuals. It reduces transmission through the sympathetic ganglia, decreasing electrically stimulated contractile responses in feline nictitating membrane.
(Enamine Bioactive Compounds)
DESCRIPTION
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
17
BOC Sciences Bioactive Compounds
Cayman Chemical Bioactives
ChEMBL Drugs
Drug Repurposing Hub
DrugCentral
DrugCentral Approved Drugs
DrugMAP
DrugMatrix
Enamine Bioactive Compounds
Enamine BioReference Compounds
Ki Database
MedChem Express Bioactive Compound Library
NPC Screening Collection
Prestwick Chemical Library
ReFrame library
Selleckchem Bioactive Compound Library
TargetMol Bioactive Compound Library
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
36
Molecular Weight
267.16
Hydrogen Bond Acceptors
2
Hydrogen Bond Donors
2
Rotatable Bonds
3
Ring Count
3
Aromatic Ring Count
2
cLogP
2.92
TPSA
32.26
Fraction CSP3
0.33
Chiral centers
0.0
Largest ring
6.0
QED
0.9
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Target
5-HT
HRH1
Histamine Receptor
5-HT Receptor
MOA
Histamine Receptor antagonist
Pathway
GPCR/G protein
Immunology/Inflammation
Neuronal Signaling
Neuroscience
Source data
