General
Preferred name
FENOTEROL
Synonyms
FENOTEROL HYDROBROMIDE ()
Fenoterol bromide ()
fenoterol, NIH ()
Fenoterol (hydrobromide) ()
Th-1165 ()
Phenoterol ()
Th-1165a ()
Phenoterol (hydrobromide) ()
Phenoterol hydrobromide ()
Fenoterol (hydrobromide) ()
FENOTEROL HBR ()
Berodual N ()
Berotec 100 ()
Berotec 200 ()
NSC-757811 ()
TH-1165A FREE BASE ()
Berodual ()
Partusisten ()
Dosberotec ()
TH 1165A ()
TH 1165A FREE BASE ()
Berotec ()
Duovent ()
TH 1165A [AS HYDROBROMIDE SALT] ()
Airum ()
P&D ID
PD009923
CAS
1944-12-3
13392-18-2
Tags
available
drug
First approval
1965
Drug indication
Airway obstruction
Asthma
Drug Status
approved
withdrawn
investigational
Max Phase
4.0
Structure
Probe scores
P&D probe-likeness score
[[ v.score ]]%
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
PRICE 29
DESCRIPTION Fenoterol hydrobromide (Th-1165a), a sympathomimetic agent, is a selective and orally active ¦Â2-adrenoceptor agonist. Fenoterol hydrobromide is an effective bronchodilator and can be used for bronchospasm associated with asthma, bronchitis and other obstructive airway diseases research[1][2].
DESCRIPTION Fenoterol hydrobromide is an orally active and selective ??2-adrenoceptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.
DESCRIPTION Fenoterol is a short-acting β2-adrenoceptor agonist (sympathomimetic) drug. The clinically used drug is a racemic mixture of enantiomers. We show the structure without specified stereochemistry to represent the mixture. The (S,R) and (R,S) enantiomers are much less active tha the (S,S) and (R,R) enantiomers. (GtoPdb)
DESCRIPTION Fenoterol (Th-1165), a sympathomimetic agent, is a selective and orally active ¦Â2-adrenoceptor agonist. Fenoterol is an effective bronchodilator and can be used for bronchospasm associated with asthma, bronchitis and other obstructive airway diseases research[1][2].
PRICE 56
DESCRIPTION Fenoterol is an agonist of ??2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
DESCRIPTION Beta2-adrenoceptor agonist; bronchodilator (LOPAC library)
DESCRIPTION Fenoterol hydrobromide is an orally active and selective β2-adrenoceptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis. (TargetMol Bioactive Compound Library)
Compound Sets
26
Cayman Chemical Bioactives
21293
ChEMBL Approved Drugs
CHEMBL32800
ChEMBL Drugs
CHEMBL32800
Concise Guide to Pharmacology 2017/18
557
Concise Guide to Pharmacology 2019/20
557
Concise Guide to Pharmacology 2021/22
557
Concise Guide to Pharmacology 2023/24
557
DrugBank
DB01288
DrugBank Approved Drugs
DB01288
DrugCentral
1155
DrugCentral Approved Drugs
1155
DrugMAP
DMIP3ZV
DrugMAP Approved Drugs
DMIP3ZV
DrugMatrix
Guide to Pharmacology
557
Ki Database
Fenoterol
LOPAC library
LSP-MoA library (Laboratory of Systems Pharmacology)
CHEMBL32800
MedChem Express Bioactive Compound Library
HY-B0976A
HY-B0976
NPC Screening Collection
Prestwick Chemical Library
ReFrame library
Selleckchem Bioactive Compound Library
fenoterol-hydrobromide
fenoterol
TargetMol Bioactive Compound Library
T22331
The Spectrum Collection
Withdrawn 2.0
w85
External IDs
42
Properties
(calculated by RDKit )
Molecular Weight
303.15
Hydrogen Bond Acceptors
5
Hydrogen Bond Donors
5
Rotatable Bonds
6
Ring Count
2
Aromatic Ring Count
2
cLogP
2.06
TPSA
92.95
Fraction CSP3
0.29
Chiral centers
2.0
Largest ring
6.0
QED
0.56
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Selectivity
beta2
Target
β2-adrenoceptor
Adrenergic Receptor
ATC
G02CA03
R03AC04
Toxicity type
cardiovascular
Pathway
GPCR/G protein
Neuroscience
Neuronal Signaling
Therapeutic Class
Bronchodilator Agents
Source data