General
Preferred name
Cefapirin
Synonyms
CEPHAPIRIN SODIUM ()
Cephapirin ()
CEPHAPIRIN ()
Cefapirin Sodium ()
CEPHAPIRIN BENZATHINE ()
BL-P 1322 ()
Cephapirin sodium salt ()
Sodium Cefapirin ()
Cefadyl ()
BL-P-1322 ()
NSC-179171 ()
Cefapirina ()
Cefapirine ()
Cefapirin benzathine ()
Metricure ()
Cephapirin compd with n,n'-dibenzylethylenediamine ()
P&D ID
PD009785
CAS
24356-60-3
21593-23-7
97468-37-6
Tags
available
drug
drug candidate
Approved by
FDA
First approval
1974
Drug indication
bacterial disease
Sepsis
Drug Status
withdrawn
vet_approved
approved
Max Phase
4.0
Probe control
Probe control not defined
Orthogonal probes
0
No orthogonal probes found
Similar probes
0
No structurally similar probes found
Structure
P&D probe-likeness score
Structure formats
[[ format ]]
[[ compound[format === 'MOL' ? 'molblock' : format.toLowerCase()] ]]
Description
(extracted from source data)
PRICE
29
DESCRIPTION
Cefapirin is a semisynthetic, first generation cephalosporin belonging to the β-lactam class of antibacterial compounds .
(GtoPdb)
DESCRIPTION
Cephapirin Benzathine is the benzathine salt form of cephapirin. Cephapirin Benzathine is the first generation cephalosporin with broad spectrum antibiotic activity[1].
DESCRIPTION
Cephalosporin C antibiotic; interferes with cell wall synthesis
(LOPAC library)
DESCRIPTION
Cefapirin sodium is the sodium salt of Cephapirin, an antimicrobial agent.
(TargetMol Bioactive Compound Library)
[[ p.pathway_name ]]
[[ compound.targets[tid].gene_name ]]
Compound Sets
21
Cayman Chemical Bioactives
ChEMBL Approved Drugs
ChEMBL Drugs
Drug Repurposing Hub
DrugBank
DrugBank Approved Drugs
DrugCentral
DrugCentral Approved Drugs
DrugMAP
DrugMAP Approved Drugs
Enamine Bioactive Compounds
Guide to Pharmacology
LOPAC library
LSP-MoA library (Laboratory of Systems Pharmacology)
MedChem Express Bioactive Compound Library
NPC Screening Collection
ReFrame library
Selleckchem Bioactive Compound Library
TargetMol Bioactive Compound Library
The Spectrum Collection
Withdrawn 2.0
[[ a.name ]]
[[ ligand_id ]]
free of charge
External IDs
83
Molecular Weight
423.06
Hydrogen Bond Acceptors
8
Hydrogen Bond Donors
2
Rotatable Bonds
7
Ring Count
3
Aromatic Ring Count
1
cLogP
0.48
TPSA
125.9
Fraction CSP3
0.35
Chiral centers
2.0
Largest ring
6.0
QED
0.37
Structural alerts
0
No structural alerts detected
Related compounds
Custom attributes
(extracted from source data)
Selectivity
Cell wall synthesis
Target
Antibacterial
antibiotic
Bacterial
Antibiotics,Bacterial
Indication
mastitis
MOA
bacterial cell wall synthesis inhibitor
ATC
J01DB08
Pathway
Microbiology/virology
Anti-infection
Therapeutic Class
Antibiotics
Source data
